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Jui-I Chao Selected Research

7- chloro- 6- piperidin- 1- ylquinoline- 5,8- dione

4/20117-Chloro-6-piperidin-1-yl-quinoline-5,8-dione (PT-262), a novel ROCK inhibitor blocks cytoskeleton function and cell migration.
10/20087-Chloro-6-piperidin-1-yl-quinoline-5,8-dione (PT-262), a novel synthetic compound induces lung carcinoma cell death associated with inhibiting ERK and CDC2 phosphorylation via a p53-independent pathway.

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Jui-I Chao Research Topics

Disease

26Neoplasms (Cancer)
11/2021 - 05/2004
10Colorectal Neoplasms (Colorectal Cancer)
01/2017 - 01/2006
7Carcinoma (Carcinomatosis)
04/2011 - 04/2004
5Lung Neoplasms (Lung Cancer)
11/2021 - 10/2008
5Breast Neoplasms (Breast Cancer)
01/2019 - 08/2012
4Carcinogenesis
09/2014 - 03/2006
3Colonic Neoplasms (Colon Cancer)
04/2013 - 09/2005
2Mitochondrial Diseases (Mitochondrial Disease)
12/2013 - 04/2013
2Urinary Bladder Neoplasms (Bladder Cancer)
04/2013 - 11/2007
2Genomic Instability
10/2010 - 12/2007
1Pleural Effusion (Pleural Effusions)
11/2021
1Non-Small-Cell Lung Carcinoma (Carcinoma, Non-Small Cell Lung)
11/2021
1Triple Negative Breast Neoplasms
01/2019
1Neoplasm Metastasis (Metastasis)
03/2016
1Embryonal Carcinoma
05/2014
1Skin Neoplasms (Skin Cancer)
04/2013
1Lymphatic Metastasis
08/2012
1Acute Promyelocytic Leukemia
03/2006
1Multiple Myeloma
03/2006
1Chromosomal Instability (Chromosome Stability)
03/2006
1Cardiovascular Diseases (Cardiovascular Disease)
03/2006

Drug/Important Bio-Agent (IBA)

16Proteins (Proteins, Gene)FDA Link
11/2021 - 05/2004
10SurvivinIBA
11/2021 - 05/2004
9SecurinIBA
09/2014 - 01/2006
6NanodiamondsIBA
01/2019 - 09/2009
6Pharmaceutical PreparationsIBA
01/2019 - 12/2006
6p38 Mitogen-Activated Protein KinasesIBA
12/2013 - 04/2004
4Oxaliplatin (Eloxatin)FDA LinkGeneric
12/2010 - 09/2005
3ErbB Receptors (EGF Receptor)IBA
11/2021 - 04/2013
3Phosphotransferases (Kinase)IBA
11/2021 - 11/2007
3Caspase 3 (Caspase-3)IBA
11/2021 - 04/2013
3Paclitaxel (Taxol)FDA LinkGeneric
01/2019 - 08/2010
3CarbonIBA
01/2017 - 08/2010
3Celecoxib (Celebrex)FDA Link
10/2008 - 09/2005
2Tyrosine Kinase InhibitorsIBA
11/2021 - 04/2013
2Gefitinib (Iressa)FDA Link
11/2021 - 04/2013
2Cetuximab (Erbitux)FDA Link
01/2019 - 01/2017
2Proteasome Endopeptidase Complex (Proteasome)IBA
01/2012 - 12/2010
27- chloro- 6- piperidin- 1- ylquinoline- 5,8- dioneIBA
04/2011 - 10/2008
2baicaleinIBA
10/2010 - 11/2007
2Small Interfering RNA (siRNA)IBA
10/2008 - 01/2006
2QuercetinIBA
11/2007 - 12/2004
2FlavonoidsIBA
11/2007 - 12/2004
2Nitric Oxide (Nitrogen Monoxide)FDA Link
05/2004 - 04/2004
1EGFR inhibitor SP101IBA
11/2021
1Epidermal Growth Factor (EGF)IBA
01/2019
1Estrogen ReceptorsIBA
01/2019
1Progesterone Receptors (Progesterone Receptor)IBA
01/2019
1Monoclonal AntibodiesIBA
01/2017
1Erlotinib Hydrochloride (CP 358,774)FDA Link
01/2017
1ClaudinsIBA
03/2016
1Tight Junction ProteinsIBA
03/2016
1honokiolIBA
11/2014
1Green Fluorescent ProteinsIBA
11/2014
1Histones (Histone)IBA
09/2014
1buteinIBA
09/2014
1Reactive Oxygen Species (Oxygen Radicals)IBA
12/2013
1Vitamin K 3 (Menadione)FDA Link
12/2013
1Acetylcysteine (Siran)FDA LinkGeneric
12/2013
1Poly(ADP-ribose) Polymerases (Poly ADP Ribose Polymerase)IBA
04/2013
1Cytochromes c (Cytochrome c)IBA
04/2013
1CateninsIBA
08/2012
1VimentinIBA
08/2012
1Biomarkers (Surrogate Marker)IBA
08/2012
1Cyclin D1IBA
08/2012
1MicroRNAs (MicroRNA)IBA
08/2012
1Protein Kinases (Protein Kinase)IBA
01/2012
1Growth Factor ReceptorsIBA
01/2012
1benzyloxycarbonylleucyl-leucyl-leucine aldehydeIBA
12/2010
1Proteasome InhibitorsIBA
12/2010
1PlatinumIBA
12/2010
14- (4- fluorophenyl)- 2- (4- hydroxyphenyl)- 5- (4- pyridyl)imidazoleIBA
12/2010
1CaspasesIBA
10/2008
12- (2- amino- 3- methoxyphenyl)- 4H- 1- benzopyran- 4- oneIBA
10/2008
1DNA (Deoxyribonucleic Acid)IBA
06/2008
1Rutin (Rutoside)IBA
11/2007
1Catechin (Z 7300)IBA
11/2007
1GenisteinIBA
11/2007
1baicalinIBA
11/2007
1arseniteIBA
03/2006
1ArsenicIBA
03/2006
1Antineoplastic Agents (Antineoplastics)IBA
03/2006
1Cytochalasin BIBA
01/2006
1Cyclooxygenase 2 Inhibitors (COX-2 Inhibitors)IBA
09/2005
1Cyclooxygenase 2 (Cyclooxygenase-2)IBA
09/2005
1Cisplatin (Platino)FDA LinkGeneric
09/2005
1Etodolac (Lodine)FDA LinkGeneric
09/2005

Therapy/Procedure

5Therapeutics
11/2021 - 08/2010
2Aftercare (After-Treatment)
11/2014 - 12/2010
1Lasers (Laser)
05/2008
1Chemoprevention
09/2005